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Ashraf Khalil
Ashraf Khalil
Professor of Medicinal Chemistry, Qatar University
Verified email at qu.edu.qa
Title
Cited by
Cited by
Year
Demonstration of isoleucine 199 as a structural determinant for the selective inhibition of human monoamine oxidase B by specific reversible inhibitors
F Hubálek, C Binda, A Khalil, M Li, A Mattevi, N Castagnoli, ...
Journal of biological chemistry 280 (16), 15761-15766, 2005
2622005
Isolation and characterization of a monoamine oxidase inhibitor from tobacco leaves
AA Khalil, S Steyn, N Castagnoli
Chemical research in toxicology 13 (1), 31-35, 2000
1182000
Design and synthesis of novel chalcones as potent selective monoamine oxidase-B inhibitors
AK • Arwa Hammuda, Raed Shalaby, Stefano Rovida, Dale E. Edmondson, Claudia ...
European Journal of Medicinal Chemistry 114, 162-169, 2016
922016
Substituted Quinazolines, Part 2. Synthesis and In‐Vitro Anticancer Evaluation of New 2‐Substituted Mercapto‐3H‐quinazoline Analogs
AA Khalil, SGA Hamide, AM Al‐Obaid, HI El‐Subbagh
Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2003
752003
Purification and characterization of 0-amylase from
AF Afifi, EA Kamel, AA Khalil, M Fawzi, MM Housery
Glob. J. Biotechnol. Biochem 3 (1), 14-21, 2008
632008
Isolation and characterization of a monoamine oxidase B selective inhibitor from tobacco smoke
AA Khalil, B Davies, N Castagnoli Jr
Bioorganic & medicinal chemistry 14 (10), 3392-3398, 2006
632006
Studies on the interactions of tobacco leaf and tobacco smoke constituents and monoamine oxidase
K Castagnoli, SJ Steyn, G Magnin, CJ Van Der Schyf, I Fourie, A Khalil, ...
Neurotoxicity research 4, 151-160, 2002
522002
SAR and molecular mechanism studies of monoamine oxidase inhibition by selected chalcone analogs
R Shalaby, JP Petzer, A Petzer, UM Ashraf, E Atari, F Alasmari, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 34 (1), 863-876, 2019
492019
Design, synthesis, and validation of novel nitrogen-based chalcone analogs against triple negative breast cancer
D Elkhalifa, AB Siddique, M Qusa, F Cyprian, K El Sayed, F Alali, ...
European Journal of Medicinal Chemistry 187, 111954, 2020
382020
Semisynthetic studies on the manzamine alkaloids
KAE Sayed, AA Khalil, M Yousaf, G Labadie, GM Kumar, SG Franzblau, ...
Journal of natural products 71 (3), 300-308, 2008
382008
Monoamine oxidase inhibitors extracted from tobacco smoke as neuroprotective factors for potential treatment of Parkinson’s disease
Y Sari, A Khalil
CNS & Neurological Disorders - Drug Targets 14 (6), 777-785, 2015
322015
Substituted Quinazolines. Part 1. Synthesis and Antitumor Activity of Certain Substituted 2‐Mercapto‐4 (3H)‐quinazolinone Analogues.
SGA Hamid, HA El‐Obeid, KA Al‐Rashood, AA Khalil, HI El‐Subbagh
ChemInform 33 (20), no-no, 2002
242002
Structure–activity relationship investigation of methoxy substitution on anticancer pyrimido[4,5-c]quinolin-1(2H)-ones
K Metwally, A Khalil, A Sallam, H Pratsinis, D Kletsas, K El Sayed
Medicinal Chemistry Research 22, 4481-4491, 2013
192013
Structure–activity relationship of piperine and its synthetic amide analogs for therapeutic potential to prevent experimentally induced ER stress in vitro
AS Hammad, S Ravindran, A Khalil, S Munusamy
Cell Stress and Chaperones 22 (3), 417-428, 2017
172017
Targeting triple negative breast cancer heterogeneity with chalcones: a molecular insight
D Elkhalifa, F Alali, AE Al Moustafa, A Khalil
Journal of drug targeting 27 (8), 830-838, 2019
152019
A novel and selective monoamine oxidase B substrate
JM Rimoldi, SG Puppali, E Isin, P Bissel, A Khalil, N Castagnoli Jr
Bioorganic & medicinal chemistry 13 (20), 5808-5813, 2005
142005
Substituted Quinazolines, 1. Synthesis and antitumor activity of certain substituted 2-mercapto-4 (3H)-quinazolinone analogs
SG Abdel Hamid, HA El-Obeid, KA Al-Rashood, AA Khalil, HI El-Subbagh
Scientia Pharmaceutica 69 (4), 351-366, 2001
132001
Concentration‐Dependent Variation of 1H‐NMR Chemical Shifts of Aromatic Protons in Sampangine Derivatives
I Katsuyama, AA Khalil, C Dunbar, JK Zjawiony
Spectroscopy letters 36 (5-6), 477-485, 2003
112003
Stereochemical studies on the novel monoamine oxidase B substrates (1R, 6S)-and (1S, 6R)-3-methyl-6-phenyl-3-aza-bicyclo [4.1. 0] heptane
P Bissel, A Khalil, JM Rimoldi, K Igarashi, D Edmondson, A Miller, ...
Bioorganic & medicinal chemistry 16 (7), 3557-3564, 2008
102008
Dipyridamole: comprehensive profile
A Khalil, F Belal, AA Al-Badr
Profiles of Drug Substances, Excipients and Related Methodology 31, 215-280, 2005
102005
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Articles 1–20