| Novel coumarin-6-sulfonamides as apoptotic anti-proliferative agents: synthesis, in vitro biological evaluation, and QSAR studies A Sabt, OM Abdelhafez, RS El-Haggar, HMF Madkour, WM Eldehna, ... Journal of enzyme inhibition and medicinal chemistry 33 (1), 1095-1107, 2018 | 100 | 2018 |
| Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC … WM Eldehna, MF Abo-Ashour, A Nocentini, RS El-Haggar, S Bua, ... European journal of medicinal chemistry 162, 147-160, 2019 | 88 | 2019 |
| Development of isatin-thiazolo [3, 2-a] benzimidazole hybrids as novel CDK2 inhibitors with potent in vitro apoptotic anti-proliferative activity: Synthesis, biological and … WM Eldehna, MA El Hassab, MF Abo-Ashour, T Al-Warhi, MM Elaasser, ... Bioorganic Chemistry 110, 104748, 2021 | 63 | 2021 |
| Anti-inflammatory screening and molecular modeling of some novel coumarin derivatives R El-Haggar, RI Al-Wabli Molecules 20 (4), 5374-5391, 2015 | 53 | 2015 |
| 3-Methylthiazolo [3, 2-a] benzimidazole-benzenesulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: Design, synthesis, biological and … AAM Alkhaldi, MM Al-Sanea, A Nocentini, WM Eldehna, ZM Elsayed, ... European Journal of Medicinal Chemistry 207, 112745, 2020 | 51 | 2020 |
| Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D … A Petreni, A Bonardi, C Lomelino, SM Osman, ZA ALOthman, ... European Journal of Medicinal Chemistry 190, 112112, 2020 | 48 | 2020 |
| Novel piperazine–chalcone hybrids and related pyrazoline analogues targeting VEGFR-2 kinase; design, synthesis, molecular docking studies, and anticancer evaluation MF Ahmed, EY Santali, R El-Haggar Journal of enzyme inhibition and medicinal chemistry 36 (1), 308-319, 2021 | 46 | 2021 |
| Development of novel benzofuran-isatin conjugates as potential antiproliferative agents with apoptosis inducing mechanism in Colon cancer WM Eldehna, R Salem, ZM Elsayed, T Al-Warhi, HR Knany, RR Ayyad, ... Journal of Enzyme Inhibition and Medicinal Chemistry 36 (1), 1423-1434, 2021 | 25 | 2021 |
| Development of pyridazine derivatives as potential EGFR inhibitors and apoptosis inducers: Design, synthesis, anticancer evaluation, and molecular modeling studies MF Ahmed, EY Santali, EMM El-Deen, IA Naguib, R El-Haggar Bioorganic Chemistry 106, 104473, 2021 | 18 | 2021 |
| Development of 2-oxindolin-3-ylidene-indole-3-carbohydrazide derivatives as novel apoptotic and anti-proliferative agents towards colorectal cancer cells WM Eldehna, MF Abo-Ashour, T Al-Warhi, ST Al-Rashood, A Alharbi, ... Journal of Enzyme Inhibition and Medicinal Chemistry 36 (1), 320-329, 2021 | 16 | 2021 |
| Fenticonazole nitrate loaded trans-novasomes for effective management of tinea corporis: design characterization, in silico study, and exploratory clinical appraisal R Albash, MH Ragaie, MAE Hassab, R El-Haggar, WM Eldehna, ... Drug Delivery 29 (1), 1100-1111, 2022 | 14 | 2022 |
| Molecular design of small organic molecules based on structural information for a conformationally constrained peptide that binds to G-CSF receptor R El-Haggar, K Kamikawa, K Machi, Z Ye, Y Ishino, T Tsumuraya, I Fujii Bioorganic & medicinal chemistry letters 20 (3), 1169-1172, 2010 | 12 | 2010 |
| Design, synthesis, molecular modeling and biological evaluation of novel Benzoxazole-Benzamide conjugates via a 2-Thioacetamido linker as potential anti … IH Eissa, R El-Haggar, MA Dahab, MF Ahmed, HA Mahdy, RI Alsantali, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1587-1599, 2022 | 10 | 2022 |
| Salmeterol xinafoate MM Anwar, RS El-Haggar, WA Zaghary Profiles of Drug Substances, Excipients and Related Methodology 40, 321-369, 2015 | 10 | 2015 |
| Synthesis, evaluation and molecular docking studies for the anti-inflammatory activity of novel 8-substituted-7-benzoyloxy-4-methyl-6-nitrocoumarin derivatives R El-Haggar, OA Abdel-Rasheed, T Nasr, HI Ali, A Goudah, N Abotaleb Afr. J. Pharm. Pharmacol 8 (48), 1213-1227, 2014 | 8 | 2014 |
| Introducing of potent cytotoxic novel 2-(aroylamino) cinnamamide derivatives against colon cancer mediated by dual apoptotic signal activation and oxidative stress AM Omar, ME El-Araby, TM Abdelghany, MK Safo, MH Ahmed, ... Bioorganic Chemistry 101, 103953, 2020 | 6 | 2020 |
| 3-Substituted-2, 3-dihydrothiazole as a promising scaffold to design EGFR inhibitors R El-Haggar, SF Hammad, RI Alsantali, MM Alrooqi, MA El Hassab, ... Bioorganic Chemistry 129, 106172, 2022 | 5 | 2022 |
| 2, 4-Diaryl-pyrimido [1, 2-a] benzimidazole derivatives as novel anticancer agents endowed with potent anti-leukemia activity: Synthesis, biological evaluation and kinase profiling MA Shaldam, D Hendrychová, R El-Haggar, V Vojáčková, TA Majrashi, ... European Journal of Medicinal Chemistry 258, 115610, 2023 | 4 | 2023 |
| Synthesis, In-vivo and In-vitro Anti-inflammatory Evaluation of some Novel Coumarin Derivatives R Al-Wabli, M Fouad, R El-Haggar Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry (Formerly …, 2018 | 4 | 2018 |
| EEDAM El-Khrisy, MA Abdel-Rahman and LA Rashed A Sabt, OM Abdelhafez, RS El-Haggar, HMF Madkour, WM Eldehna J. Enzyme Inhib. Med. Chem 33, 1095-1107, 2018 | 4 | 2018 |
