| Design, synthesis, biological evaluation and docking studies of new 3-(4, 5-dihydro-1H-pyrazol/isoxazol-5-yl)-2-phenyl-1H-indole derivatives as potent antioxidants and 15 … HS ElBordiny, MM El-Miligy, SE Kassab, H Daabees, WAM Ali, ... European journal of medicinal chemistry 145, 594-605, 2018 | 47 | 2018 |
| Discovery of new indomethacin-based analogs with potentially selective cyclooxygenase-2 inhibition and observed diminishing to PGE2 activities SE Kassab, MA Khedr, HI Ali, MM Abdalla European journal of medicinal chemistry 141, 306-321, 2017 | 34 | 2017 |
| Design, synthesis, 3D pharmacophore, QSAR, and docking studies of carboxylic acid derivatives as Histone Deacetylase inhibitors and cytotoxic agents MM Abdel-Atty, NA Farag, SE Kassab, RAT Serya, KAM Abouzid Bioorganic Chemistry 57, 65-82, 2014 | 33 | 2014 |
| Synthesis of 1H-Indole-2,3-Dione-3-Thiosemicarbazone Ribonucleosides as Antibacterial Agents SE Kassab, GH Hegazy, NM Eid, KM Amin, AA El-Gendy Nucleosides, Nucleotides and Nucleic Acids 29 (1), 72-80, 2010 | 29 | 2010 |
| Base-catalyzed one-step synthesis of 5, 7-disubstituted-1, 2, 4-triazolo [1, 5-a] pyrimidines X He, SE Kassab, G Heinzl, F Xue Tetrahedron letters 56 (8), 1034-1037, 2015 | 25 | 2015 |
| A promising anti-cancer and anti-oxidant agents based on the pyrrole and fused pyrrole: synthesis, docking studies and biological evaluation S Said Fatahala, E Ahmed Shalaby, S Emam Kassab, M Said Mohamed Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2015 | 21 | 2015 |
| Design, synthesis and biological evaluation of novel thiohydantoin derivatives as antiproliferative agents: A combined experimental and theoretical assessments MM Elbadawi, AI Khodair, MK Awad, SE Kassab, MT Elsaady, ... Journal of Molecular Structure 1249, 131574, 2022 | 16 | 2022 |
| Febuxostat-based amides and some derived heterocycles targeting xanthine oxidase and COX inhibition. Synthesis, in vitro and in vivo biological evaluation, molecular modeling … AY Rashad, SE Kassab, HG Daabees, AEA Moneim, SAF Rostom Bioorganic Chemistry 113, 104948, 2021 | 12 | 2021 |
| Synthesis of novel d-α-galactopyranosyl-l-seryl/l-threonyl-l-alanyl-l-alanine as useful precursors of new glycopeptide antibiotics with computational calculations studies AI Khodair, SE Kassab, NA Kheder, AM Fahim Carbohydrate Research 514, 108546, 2022 | 11 | 2022 |
| Structure-based design generated novel hydroxamic acid based preferential HDAC6 lead inhibitor with on-target cytotoxic activity against primary choroid plexus carcinoma SE Kassab, S Mowafy, AM Alserw, JA Seliem, SM El-Naggar, NN Omar, ... Journal of enzyme inhibition and medicinal chemistry 34 (1), 1062-1077, 2019 | 11 | 2019 |
| Anti-Cancer Agents Med SS Fatahala, EA Shalaby, SE Kassab, MS Mohamed Chem 15, 517-526, 2015 | 9 | 2015 |
| Rational design of biodegradable sulphonamide candidates treating septicaemia by synergistic dual inhibition of COX-2/PGE2 axis and DHPS enzyme NH El-Dershaby, SA El-Hawash, SE Kassab, HG Dabees, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1737-1751, 2022 | 6 | 2022 |
| Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity MA Ragab, M Elagawany, H Daabees, ASF Ahmed, EM Awad, C Billon, ... Bioorganic Chemistry 119, 105554, 2022 | 5 | 2022 |
| Indomethacin from Anti-Inflammatory to Anticancer Agent SE Kassab Medicinal Chemistry, 2018 | 4 | 2018 |
| Structural Basis of Selective Human Indoleamine‐2, 3‐dioxygenase 1 (hIDO1) Inhibition SE Kassab, S Mowafy ChemMedChem 16 (20), 3149-3164, 2021 | 3 | 2021 |
| Rational design and synthesis of new selective COX-2 inhibitors with In Vivo PGE2-lowering activity by tethering benzenesulfonamide and 1, 2, 3-triazole pharmacophores to some … NH El-Dershaby, SA El-Hawash, SE Kassab, HG Daabees, ... Pharmaceuticals 15 (10), 1165, 2022 | 2 | 2022 |
| CORRIGENDUM A Promising Anti-Cancer and Anti-Oxidant Agents Based on the Pyrrole and Fused Pyrrole: Synthesis, Docking Studies and Biological Evaluation SS Fatahala, EA Shalaby, SE Kassab Anti-cancer agents in medicinal chemistry 18 (10), 1505, 2018 | 2 | 2018 |
| Synthesis of New 9-glycosyl-4, 9-dihydropyrano [3, 4-b] indole-1 (3 H)-ones as Antibacterial Agents SE Kassab, GH Hegazy, NM Eid, KM Amin, AA El-Gendy Nucleosides, Nucleotides and Nucleic Acids 30 (11), 991-998, 2011 | 2 | 2011 |
| Camptothecin structure simplification elaborated new imidazo [2, 1-b] quinazoline derivative as a human topoisomerase I inhibitor with efficacy against bone cancer cells and … AI Khodair, SM El-Hallouty, B Cagle-White, MHA Aziz, MK Hanafy, ... European Journal of Medicinal Chemistry 265, 116049, 2024 | | 2024 |
| Molecular-based design, synthesis and docking studies of new benzimidazole derivatives as potential bacterial peptide deformylase inhibitors S Kassab ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 254, 2017 | | 2017 |
