| Boron-containing enamine and enamide linchpins in the synthesis of nitrogen heterocycles JD St. Denis, A Zajdlik, J Tan, P Trinchera, CF Lee, Z He, S Adachi, ... Journal of the American Chemical Society 136 (50), 17669-17673, 2014 | 70 | 2014 |
| Photocatalytic reverse polarity Povarov reaction JA Leitch, ALF de Arriba, J Tan, O Hoff, CM Martínez, DJ Dixon Chemical Science 9 (32), 6653-6658, 2018 | 59 | 2018 |
| Multicomponent mapping of boron chemotypes furnishes selective enzyme inhibitors J Tan, AB Cognetta III, DB Diaz, KM Lum, S Adachi, S Kundu, BF Cravatt, ... Nature communications 8 (1), 1760, 2017 | 47 | 2017 |
| De Novo design of boron-based peptidomimetics as potent inhibitors of human ClpP in the presence of human ClpX J Tan, JJ Grouleff, Y Jitkova, DB Diaz, EC Griffith, W Shao, ... Journal of Medicinal Chemistry 62 (13), 6377-6390, 2019 | 37 | 2019 |
| Mechanistic investigation of aziridine aldehyde-driven peptide macrocyclization: the imidoanhydride pathway S Zaretsky, JL Hickey, J Tan, D Pichugin, MAS Denis, S Ler, BKW Chung, ... Chemical science 6 (10), 5446-5455, 2015 | 29 | 2015 |
| Rational design of calpain inhibitors based on calpastatin peptidomimetics KE Low, S Ler, KJ Chen, RL Campbell, JL Hickey, J Tan, CCG Scully, ... Journal of Medicinal Chemistry 59 (11), 5403-5415, 2016 | 24 | 2016 |
| Synthesis, characterization and radiolabeling of carborane-functionalized tetrazines for use in inverse electron demand Diels–Alder ligation reactions AR Genady, J Tan, E Mohamed, A Zlitni, N Janzen, JF Valliant Journal of Organometallic Chemistry 791, 204-213, 2015 | 24 | 2015 |
| Borylated reagents for multicomponent reactions J Tan, AK Yudin Drug Discovery Today: Technologies 29, 51-60, 2018 | 20 | 2018 |
| Twisted amide electrophiles enable cyclic peptide sequencing S Zaretsky, V Rai, G Gish, MW Forbes, M Kofler, CY Joy, J Tan, JL Hickey, ... Organic & Biomolecular Chemistry 13 (27), 7384-7388, 2015 | 11 | 2015 |
| Macrocyclic templates for library synthesis of peptido-conjugates S Zaretsky, J Tan, JL Hickey, AK Yudin Peptide Libraries: Methods and Protocols, 67-80, 2015 | 9 | 2015 |
| Towards depeptidized aminoboronic acid derivatives through the use of borylated iminium ions V Trudel, C Brien, J Tan, AK Yudin Chemical Communications 58 (32), 5033-5036, 2022 | 4 | 2022 |
| An Exploration of Regioselectivity During Formation of Aminoboronates from Epoxides A Trofimova, C Brien, J Tan, V Trudel Synlett, 2024 | | 2024 |
| Polo like kinase 4 inhibitors C Ndubaku, JT Moore, PA Gibbons, JH Chang, FA Romero, X Du, ... US Patent 11,858,915, 2024 | | 2024 |
| Pyrido[3,2-d]pyrimidine compounds uses thereof for treating a proliferative disease PL Beaulieu, E Beaulieu, S Tripathy, E Benoit, J Tan, H Lavoie, Y Rose, ... WO Patent 2022221939 A1, 2022 | | 2022 |
