Targeting tumor hypoxia: suppression of breast tumor growth and metastasis by novel carbonic anhydrase IX inhibitors Y Lou, PC McDonald, A Oloumi, S Chia, C Ostlund, A Ahmadi, A Kyle, ... Cancer research 71 (9), 3364-3376, 2011 | 784 | 2011 |
Ureido-substituted benzenesulfonamides potently inhibit carbonic anhydrase IX and show antimetastatic activity in a model of breast cancer metastasis F Pacchiano, F Carta, PC McDonald, Y Lou, D Vullo, A Scozzafava, ... Journal of medicinal chemistry 54 (6), 1896-1902, 2011 | 531 | 2011 |
Antiglaucoma carbonic anhydrase inhibitors: a patent review E Masini, F Carta, A Scozzafava, CT Supuran Expert opinion on therapeutic patents 23 (6), 705-716, 2013 | 323 | 2013 |
Diuretics with carbonic anhydrase inhibitory action: a patent and literature review (2005–2013) F Carta, CT Supuran Expert opinion on therapeutic patents 23 (6), 681-691, 2013 | 299 | 2013 |
Antiobesity carbonic anhydrase inhibitors: a literature and patent review A Scozzafava, CT Supuran, F Carta Expert opinion on therapeutic patents 23 (6), 725-735, 2013 | 290 | 2013 |
Sulfonamides: a patent review (2008–2012) F Carta, A Scozzafava, CT Supuran Expert opinion on therapeutic patents 22 (7), 747-758, 2012 | 263 | 2012 |
Dithiocarbamates strongly inhibit carbonic anhydrases and show antiglaucoma action in vivo F Carta, M Aggarwal, A Maresca, A Scozzafava, R McKenna, E Masini, ... Journal of medicinal chemistry 55 (4), 1721-1730, 2012 | 256 | 2012 |
Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: three for the price of one CT Supuran, V Alterio, A Di Fiore, K D’Ambrosio, F Carta, SM Monti, ... Medicinal Research Reviews 38 (6), 1799-1836, 2018 | 245 | 2018 |
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule F Carta, C Temperini, A Innocenti, A Scozzafava, K Kaila, CT Supuran Journal of Medicinal Chemistry 53 (15), 5511-5522, 2010 | 240 | 2010 |
Specific inhibition of carbonic anhydrase IX activity enhances the in vivo therapeutic effect of tumor irradiation L Dubois, S Peeters, NG Lieuwes, N Geusens, A Thiry, S Wigfield, F Carta, ... Radiotherapy and Oncology 99 (3), 424-431, 2011 | 212 | 2011 |
Sulfonamides and their isosters as carbonic anhydrase inhibitors F Carta, CT Supuran, A Scozzafava Future medicinal chemistry 6 (10), 1149-1165, 2014 | 204 | 2014 |
Antimetastatic effect of sulfamate carbonic anhydrase IX inhibitors in breast carcinoma xenografts RG Gieling, M Babur, L Mamnani, N Burrows, BA Telfer, F Carta, ... Journal of medicinal chemistry 55 (11), 5591-5600, 2012 | 182 | 2012 |
Design and synthesis of novel indole β-diketo acid derivatives as HIV-1 integrase inhibitors M Sechi, M Derudas, R Dallocchio, A Dessì, A Bacchi, L Sannia, F Carta, ... Journal of medicinal chemistry 47 (21), 5298-5310, 2004 | 182 | 2004 |
Dithiocarbamates: a new class of carbonic anhydrase inhibitors. Crystallographic and kinetic investigations F Carta, M Aggarwal, A Maresca, A Scozzafava, R McKenna, CT Supuran Chemical Communications 48 (13), 1868-1870, 2012 | 181 | 2012 |
Novel therapies for glaucoma: a patent review 2007–2011 F Carta, CT Supuran, A Scozzafava Expert opinion on therapeutic patents 22 (1), 79-88, 2012 | 165 | 2012 |
A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects F Carta, LDC Mannelli, M Pinard, C Ghelardini, A Scozzafava, ... Bioorganic & medicinal chemistry 23 (8), 1828-1840, 2015 | 157 | 2015 |
Carbonic anhydrase IX from cancer-associated fibroblasts drives epithelial-mesenchymal transition in prostate carcinoma cells T Fiaschi, E Giannoni, L Taddei, P Cirri, A Marini, G Pintus, C Nativi, ... Cell Cycle 12 (11), 1791-1801, 2013 | 152 | 2013 |
Dithiocarbamates strongly inhibit the β-class carbonic anhydrases from Mycobacterium tuberculosis A Maresca, F Carta, D Vullo, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 28 (2), 407-411, 2013 | 150 | 2013 |
Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment A Angeli, F Carta, A Nocentini, JY Winum, R Zalubovskis, A Akdemir, ... Metabolites 10 (10), 412, 2020 | 136 | 2020 |
[(Cp‐R)M(CO)3] (M=Re or 99mTc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX D Can, B Spingler, P Schmutz, F Mendes, P Raposinho, C Fernandes, ... Angewandte Chemie International Edition 51 (14), 3354-3357, 2012 | 133 | 2012 |