Recent advances in the therapeutic applications of pyrazolines MR Shaaban, AS Mayhoub, AM Farag Expert opinion on therapeutic patents 22 (3), 253-291, 2012 | 170 | 2012 |
Regioselective synthesis and antitumor screening of some novel N-phenylpyrazole derivatives AM Farag, AS Mayhoub, SE Barakat, AH Bayomi Bioorganic & medicinal chemistry 16 (2), 881-889, 2008 | 168 | 2008 |
Synthesis of new N-phenylpyrazole derivatives with potent antimicrobial activity AM Farag, AS Mayhoub, SE Barakat, AH Bayomi Bioorganic & medicinal chemistry 16 (8), 4569-4578, 2008 | 157 | 2008 |
Synthesis and analgesic/anti-inflammatory evaluation of fused heterocyclic ring systems incorporating phenylsulfonyl moiety MR Shaaban, TS Saleh, AS Mayhoub, A Mansour, AM Farag Bioorganic & medicinal chemistry 16 (12), 6344-6352, 2008 | 146 | 2008 |
Discovery and Characterization of Potent Thiazoles versus Methicillin- and Vancomycin-Resistant Staphylococcus aureus H Mohammad, AS Mayhoub, A Ghafoor, M Soofi, RA Alajlouni, ... Journal of medicinal chemistry 57 (4), 1609-1615, 2014 | 113 | 2014 |
Single step synthesis of new fused pyrimidine derivatives and their evaluation as potent Aurora-A kinase inhibitors MR Shaaban, TS Saleh, AS Mayhoub, AM Farag European Journal of Medicinal Chemistry 46 (9), 3690-3695, 2011 | 108 | 2011 |
Anti-biofilm activity and synergism of novel thiazole compounds with glycopeptide antibiotics against multidrug-resistant staphylococci H Mohammad, AS Mayhoub, M Cushman, MN Seleem The Journal of antibiotics 68 (4), 259-266, 2015 | 102 | 2015 |
Design, synthesis and structure–activity relationship study of novel pyrazole-based heterocycles as potential antitumor agents AM Farag, KAK Ali, TMA El-Debss, AS Mayhoub, AGE Amr, ... European journal of medicinal chemistry 45 (12), 5887-5898, 2010 | 99 | 2010 |
Synthesis and antibacterial evaluation of a novel series of synthetic phenylthiazole compounds against methicillin-resistant Staphylococcus aureus (MRSA) H Mohammad, PVN Reddy, D Monteleone, AS Mayhoub, M Cushman, ... European journal of medicinal chemistry 94, 306-316, 2015 | 95 | 2015 |
The tamoxifen metabolite norendoxifen is a potent and selective inhibitor of aromatase (CYP19) and a potential lead compound for novel therapeutic agents WJ Lu, C Xu, Z Pei, AS Mayhoub, M Cushman, DA Flockhart Breast cancer research and treatment 133, 99-109, 2012 | 90 | 2012 |
Optimizing thiadiazole analogues of resveratrol versus three chemopreventive targets AS Mayhoub, L Marler, TP Kondratyuk, EJ Park, JM Pezzuto, M Cushman Bioorganic & medicinal chemistry 20 (1), 510-520, 2012 | 80 | 2012 |
Unexpected N-acetylation of capreomycin by mycobacterial Eis enzymes JL Houghton, KD Green, RE Pricer, AS Mayhoub, S Garneau-Tsodikova Journal of antimicrobial chemotherapy 68 (4), 800-805, 2013 | 76 | 2013 |
Antibacterial characterization of novel synthetic thiazole compounds against methicillin-resistant Staphylococcus pseudintermedius H Mohammad, PVN Reddy, D Monteleone, AS Mayhoub, M Cushman, ... PloS one 10 (6), e0130385, 2015 | 69 | 2015 |
Synthesis and Structure‐Activity Relationship Studies of Pyrazole‐based Heterocycles as Antitumor Agents AM Farag, AS Mayhoub, TMA Eldebss, AGE Amr, KAK Ali, ... Archiv der Pharmazie 343 (7), 384-396, 2010 | 65 | 2010 |
Diphenylpyrroles: novel p53 activators SM Gomha, TMA Eldebss, MM Abdulla, AS Mayhoub European journal of medicinal chemistry 82, 472-479, 2014 | 62 | 2014 |
Novel 4‐heteroaryl‐antipyrines as DPP‐IV inhibitors SM Gomha, TMA Eldebss, MG Badrey, MM Abdulla, AS Mayhoub Chemical Biology & Drug Design 86 (5), 1292-1303, 2015 | 61 | 2015 |
A novel hybrid of 6-chlorotacrine and metal–amyloid-β modulator for inhibition of acetylcholinesterase and metal-induced amyloid-β aggregation A Kochi, TJ Eckroat, KD Green, AS Mayhoub, MH Lim, ... Chemical Science 4 (11), 4137-4145, 2013 | 61 | 2013 |
An investigation of phenylthiazole antiflaviviral agents AS Mayhoub, M Khaliq, C Botting, Z Li, RJ Kuhn, M Cushman Bioorganic & medicinal chemistry 19 (12), 3845-3854, 2011 | 61 | 2011 |
Second-generation phenylthiazole antibiotics with enhanced pharmacokinetic properties MA Seleem, AM Disouky, H Mohammad, TM Abdelghany, AS Mancy, ... Journal of medicinal chemistry 59 (10), 4900-4912, 2016 | 60 | 2016 |
Design, synthesis, and biological evaluation of thiazoles targeting flavivirus envelope proteins AS Mayhoub, M Khaliq, RJ Kuhn, M Cushman Journal of medicinal chemistry 54 (6), 1704-1714, 2011 | 59 | 2011 |