Department NEUROFARBA - Pharmaceutical and nutraceutical section
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Central nicotinic receptors: structure, function, ligands, and therapeutic potential
MN Romanelli, P Gratteri, L Guandalini, E Martini, C Bonaccini, F Gualtieri
ChemMedChem: Chemistry Enabling Drug Discovery 2 (6), 746-767, 2007
The crystal structure of human telomeric DNA complexed with berberine: an interesting case of stacked ligand to G-tetrad ratio higher than 1: 1
C Bazzicalupi, M Ferraroni, AR Bilia, F Scheggi, P Gratteri
Nucleic acids research 41 (1), 632-638, 2013
Novel 4/3-((4-oxo-5-(2-oxoindolin-3-ylidene) thiazolidin-2-ylidene) amino) benzenesulfonamides: Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and …
WM Eldehna, MF Abo-Ashour, A Nocentini, P Gratteri, IH Eissa, M Fares, ...
European journal of medicinal chemistry 139, 250-262, 2017
Spectroscopic, molecular modeling, and NMR-spectroscopic investigation of the binding mode of the natural alkaloids berberine and sanguinarine to human telomeric G-quadruplex DNA
I Bessi, C Bazzicalupi, C Richter, HRA Jonker, K Saxena, C Sissi, ...
ACS chemical biology 7 (6), 1109-1119, 2012
Total Syntheses of Casuarine and Its 6‐O‐α‐Glucoside: Complementary Inhibition towards Glycoside Hydrolases of the GH31 and GH37 Families
F Cardona, C Parmeggiani, E Faggi, C Bonaccini, P Gratteri, L Sim, ...
Chemistry–A European Journal 15 (7), 1627-1636, 2009
Determinants for tight and selective binding of a medicinal dicarbene gold (I) complex to a telomeric DNA G‐quadruplex: a joint ESI MS and XRD investigation
C Bazzicalupi, M Ferraroni, F Papi, L Massai, B Bertrand, L Messori, ...
Angewandte Chemie 128 (13), 4328-4331, 2016
Benzenesulfonamides incorporating flexible triazole moieties are highly effective carbonic anhydrase inhibitors: synthesis and kinetic, crystallographic, computational, and …
A Nocentini, M Ferraroni, F Carta, M Ceruso, P Gratteri, C Lanzi, E Masini, ...
Journal of Medicinal Chemistry 59 (23), 10692-10704, 2016
Enhanced curcumin permeability by SLN formulation: The PAMPA approach
C Righeschi, MC Bergonzi, B Isacchi, C Bazzicalupi, P Gratteri, AR Bilia
LWT-Food Science and Technology 66, 475-483, 2016
Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC …
WM Eldehna, MF Abo-Ashour, A Nocentini, RS El-Haggar, S Bua, ...
European journal of medicinal chemistry 162, 147-160, 2019
Sulfonamide inhibitors of human carbonic anhydrases designed through a three-tails approach: improving ligand/isoform matching and selectivity of action
A Bonardi, A Nocentini, S Bua, J Combs, C Lomelino, J Andring, ...
Journal of medicinal chemistry 63 (13), 7422-7444, 2020
A Novel Selective GABAA α1 Receptor Agonist Displaying Sedative and Anxiolytic-like Properties in Rodents
S Selleri, F Bruni, C Costagli, A Costanzo, G Guerrini, G Ciciani, P Gratteri, ...
Journal of medicinal chemistry 48 (21), 6756-6760, 2005
Experimental design in the development of voltammetric method for the assay of omeprazole
S Pinzauti, P Gratteri, S Furlanetto, P Mura, E Dreassi, R Phan-Tan-Luu
Journal of pharmaceutical and biomedical analysis 14 (8-10), 881-889, 1996
Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms
A Nocentini, A Bonardi, P Gratteri, B Cerra, A Gioiello, CT Supuran
Journal of Enzyme Inhibition and Medicinal Chemistry 33 (1), 1453-1459, 2018
Insight into 2-phenylpyrazolo [1, 5-a] pyrimidin-3-yl acetamides as peripheral benzodiazepine receptor ligands: synthesis, biological evaluation and 3D-QSAR investigation
S Selleri, P Gratteri, C Costagli, C Bonaccini, A Costanzo, F Melani, ...
Bioorganic & medicinal chemistry 13 (16), 4821-4834, 2005
3-Hydrazinoisatin-based benzenesulfonamides as novel carbonic anhydrase inhibitors endowed with anticancer activity: Synthesis, in vitro biological evaluation and in silico …
MF Abo-Ashour, WM Eldehna, A Nocentini, A Bonardi, S Bua, HS Ibrahim, ...
European Journal of Medicinal Chemistry 184, 111768, 2019
Selenols: A new class of carbonic anhydrase inhibitors
A Angeli, D Tanini, A Nocentini, A Capperucci, M Ferraroni, P Gratteri, ...
Chemical Communications 55 (5), 648-651, 2019
Deciphering the mechanism of human carbonic anhydrases inhibition with sulfocoumarins: computational and experimental studies
A Nocentini, F Carta, M Tanc, S Selleri, CT Supuran, C Bazzicalupi, ...
Chemistry–A European Journal 24 (31), 7840-7844, 2018
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the …
HS Ibrahim, HA Allam, WR Mahmoud, A Bonardi, A Nocentini, P Gratteri, ...
European Journal of Medicinal Chemistry 152, 1-9, 2018
Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and …
WM Eldehna, GH Al-Ansary, S Bua, A Nocentini, P Gratteri, A Altoukhy, ...
European Journal of Medicinal Chemistry 127, 521-530, 2017
Phosphorus versus sulfur: Discovery of benzenephosphonamidates as versatile sulfonamide‐mimic chemotypes acting as carbonic anhydrase inhibitors
A Nocentini, P Gratteri, CT Supuran
Chemistry–A European Journal 25 (5), 1188-1192, 2019
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