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Dr. Rania B. Bakr
Dr. Rania B. Bakr
Associate Professor of pharmaceutical organic chemistry, faculty of pharmacy, Beni-Suef University
Verified email at pharm.bsu.edu.eg - Homepage
Title
Cited by
Cited by
Year
Design, synthesis and biological evaluation of some novel benzothiazole/benzoxazole and/or benzimidazole derivatives incorporating a pyrazole scaffold as antiproliferative agents
MA Abdelgawad, RB Bakr, HA Omar
Bioorganic chemistry 74, 82-90, 2017
1082017
Synthesis of chalcones derivatives and their biological activities: a review
NAA Elkanzi, H Hrichi, RA Alolayan, W Derafa, FM Zahou, RB Bakr
ACS omega 7 (32), 27769-27786, 2022
1062022
Design, synthesis and antitumor activity of novel pyrazolo [3, 4-d] pyrimidine derivatives as EGFR-TK inhibitors
MA Abdelgawad, RB Bakr, OA Alkhoja, WR Mohamed
Bioorganic chemistry 66, 88-96, 2016
732016
Novel pyrimidine-pyridine hybrids: synthesis, cyclooxygenase inhibition, anti-inflammatory activity and ulcerogenic liability
MA Abdelgawad, RB Bakr, AA Azouz
Bioorganic chemistry 77, 339-348, 2018
662018
New pyrimidine-benzoxazole/benzimidazole hybrids: Synthesis, antioxidant, cytotoxic activity, in vitro cyclooxygenase and phospholipase A2-V inhibition
MA Abdelgawad, RB Bakr, W Ahmad, MM Al-Sanea, HAH Elshemy
Bioorganic chemistry 92, 103218, 2019
562019
Pyrimidine and fused pyrimidine derivatives as promising protein kinase inhibitors for cancer treatment
KRA Abdellatif, RB Bakr
Medicinal Chemistry Research 30, 31-49, 2021
532021
New advances in synthesis and clinical aspects of pyrazolo [3, 4-d] pyrimidine scaffolds
KRA Abdellatif, RB Bakr
Bioorganic chemistry 78, 341-357, 2018
532018
Synthesis and Anticancer Activity of Some New Pyrazolo[3,4-d]pyrimidin-4-one Derivatives
KRA Abdellatif, EKA Abdelall, MA Abdelgawad, RR Ahmed, RB Bakr
Molecules 19 (3), 3297-3309, 2014
502014
Synthesis, cyclooxygenase inhibition, anti-inflammatory evaluation and ulcerogenic liability of new 1-phenylpyrazolo[3,4-d]pyrimidine derivatives
RB Bakr, AA Azouz, KRA Abdellatif
Journal of enzyme inhibition and medicinal chemistry 31 (sup2), 6-12, 2016
432016
New 1, 2, 3-triazole-containing hybrids as antitumor candidates: Design, click reaction synthesis, DFT calculations, and molecular docking study
IH El Azab, HS El-Sheshtawy, RB Bakr, NAA Elkanzi
Molecules 26 (3), 708, 2021
362021
Nitric oxide-NASIDS donor prodrugs as hybrid safe anti-inflammatory agents
K RA Abdellatif, E KA Abdelall, R B Bakr
Current topics in medicinal chemistry 17 (8), 941-955, 2017
342017
Sulfonamide-based 4-anilinoquinoline derivatives as novel dual Aurora kinase (AURKA/B) inhibitors: Synthesis, biological evaluation and in silico insights
MM Al-Sanea, A Elkamhawy, S Paik, K Lee, AM El Kerdawy, BSN Abbas, ...
Bioorganic & medicinal chemistry 28 (13), 115525, 2020
312020
Selective cyclooxygenase inhibition and ulcerogenic liability of some newly prepared anti-inflammatory agents having thiazolo [4, 5-d] pyrimidine scaffold
RB Bakr, AA Ghoneim, AA Azouz
Bioorganic chemistry 88, 102964, 2019
292019
Design, Synthesis, Molecular Modeling Study, and Antimicrobial Activity of Some Novel Pyrano [2, 3‐b] pyridine and Pyrrolo [2, 3‐b] pyrano [2.3‐d] pyridine Derivatives
NAA Elkanzi, RB Bakr, AA Ghoneim
Journal of Heterocyclic Chemistry, 2019
282019
Novel phenolic compounds as potential dual EGFR and COX-2 inhibitors: Design, semisynthesis, in vitro biological evaluation and in silico Insights
MA Abdelgawad, A Musa, AH Almalki, SI Alzarea, EM Mostafa, ...
Drug design, development and therapy, 2325-2337, 2021
272021
Synthesis, EGFR Inhibition and Anti-cancer Activity of New 3, 6-dimethyl-1-phenyl-4-(substituted-methoxy) pyrazolo [3, 4-d] pyrimidine Derivatives
R B Bakr, A BM Mehany, K RA Abdellatif
Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2017
272017
Design and synthesis of new EGFR-tyrosine kinase inhibitors containing pyrazolo [3, 4-d] pyrimidine cores as anticancer agents
RB Bakr, EKA Abdelall, MK Abdel-Hamid, MM Kandeel
Bulletin of Pharmaceutical Sciences Assiut University 35 (1), 27-42, 2012
232012
Discovery of a COX-2 selective inhibitor hit with anti-inflammatory activity and gastric ulcer protective effect
MA Abdelgawad, RB Bakr, AO El-Gendy, GM Kamel, AA Azouz, ...
Future medicinal chemistry 9 (16), 1899-1912, 2017
212017
Targeting tumor cells with pyrazolo [3, 4-d] pyrimidine scaffold: A literature review on synthetic approaches, structure activity relationship, structural and target-based …
MA Abdelgawad, NAA Elkanzi, AA Nayl, A Musa, NH Alotaibi, WAA Arafa, ...
Arabian Journal of Chemistry 15 (5), 103781, 2022
202022
Preparation of some novel thiazolidinones, imidazolinones, and azetidinone bearing pyridine and pyrimidine moieties with antimicrobial activity
RB Bakr, NAA Elkanzi
Journal of heterocyclic chemistry 57 (7), 2977-2989, 2020
202020
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