Oleuropein and derivatives from olives as Tau aggregation inhibitors A Daccache, C Lion, N Sibille, M Gerard, C Slomianny, G Lippens, ... Neurochemistry international 58 (6), 700-707, 2011 | 203 | 2011 |
Design, Synthesis, and Biological Evaluation of a Series of 2-Hydroxyisoquinoline-1,3(2H,4H)-diones as Dual Inhibitors of Human Immunodeficiency Virus Type 1 … M Billamboz, F Bailly, ML Barreca, L De Luca, JF Mouscadet, C Calmels, ... Journal of medicinal chemistry 51 (24), 7717-7730, 2008 | 152 | 2008 |
Magnesium Chelating 2-Hydroxyisoquinoline-1,3(2H,4H)-diones, as Inhibitors of HIV-1 Integrase and/or the HIV-1 Reverse Transcriptase Ribonuclease H Domain … M Billamboz, F Bailly, C Lion, N Touati, H Vezin, C Calmels, ML Andréola, ... Journal of medicinal chemistry 54 (6), 1812-1824, 2011 | 149 | 2011 |
Non-photoinduced biological properties of verteporfin F Gibault, M Corvaisier, F Bailly, G Huet, P Melnyk, P Cotelle Current medicinal chemistry 23 (11), 1171-1184, 2016 | 109 | 2016 |
Reaction of rosmarinic acid with nitrite ions in acidic conditions: discovery of nitro-and dinitrorosmarinic acids as new anti-HIV-1 agents M Dubois, F Bailly, G Mbemba, JF Mouscadet, Z Debyser, M Witvrouw, ... Journal of medicinal chemistry 51 (8), 2575-2579, 2008 | 104 | 2008 |
Anti-HIV activities of natural antioxidant caffeic acid derivatives: toward an antiviral supplementation diet F Bailly, P Cotelle Frontiers in Medicinal Chemistry: Volume 4, 491-505, 2009 | 102 | 2009 |
Bistramides A, B, C, D, and K: a new class of bioactive cyclic polyethers from Lissoclinum bistratum JF Biard, C Roussakis, JM Kornprobst, D Gouiffes-Barbin, JF Verbist, ... Journal of natural products 57 (10), 1336-1345, 1994 | 98 | 1994 |
Targeting transcriptional enhanced associate domains (TEADs) miniperspective F Gibault, M Sturbaut, F Bailly, P Melnyk, P Cotelle Journal of Medicinal Chemistry 61 (12), 5057-5072, 2017 | 89 | 2017 |
Structure-activity relationships of HIV-1 integrase inhibitors-enzyme-ligand interactions C Maurin, F Bailly, P Cotelle Current medicinal chemistry 10 (18), 1795-1810, 2003 | 84 | 2003 |
Molecular features of the YAP inhibitor verteporfin: synthesis of hexasubstituted dipyrrins as potential inhibitors of YAP/TAZ, the downstream effectors of the hippo pathway F Gibault, F Bailly, M Corvaisier, M Coevoet, G Huet, P Melnyk, P Cotelle ChemMedChem 12 (12), 954-961, 2017 | 82 | 2017 |
2-Hydroxyisoquinoline-1, 3 (2H, 4H)-diones as inhibitors of HIV-1 integrase and reverse transcriptase RNase H domain: Influence of the alkylation of position 4 M Billamboz, F Bailly, C Lion, C Calmels, ML Andréola, M Witvrouw, ... European journal of medicinal chemistry 46 (2), 535-546, 2011 | 82 | 2011 |
Hepatitis B virus replication is blocked by a 2-hydroxyisoquinoline-1, 3 (2H, 4H)-dione (HID) inhibitor of the viral ribonuclease H activity CW Cai, E Lomonosova, EA Moran, X Cheng, KB Patel, F Bailly, P Cotelle, ... Antiviral research 108, 48-55, 2014 | 81 | 2014 |
Antioxidant properties of 3-hydroxycoumarin derivatives F Bailly, C Maurin, E Teissier, H Vezin, P Cotelle Bioorganic & medicinal chemistry 12 (21), 5611-5618, 2004 | 80 | 2004 |
Improved preparation and structural investigation of 4-aryl-4-oxo-2-hydroxy-2-butenoic acids and methyl esters C Maurin, F Bailly, P Cotelle Tetrahedron 60 (31), 6479-6486, 2004 | 76 | 2004 |
Patented HIV-1 integrase inhibitors (1998-2005) P Cotelle Recent Patents on Anti-Infective Drug Discovery 1 (1), 1-15, 2006 | 71 | 2006 |
4-Substituted 2-Hydroxyisoquinoline-1,3(2H,4H)-diones as a Novel Class of HIV-1 Integrase Inhibitors M Billamboz, V Suchaud, F Bailly, C Lion, J Demeulemeester, C Calmels, ... ACS Medicinal Chemistry Letters 4 (7), 606-611, 2013 | 70 | 2013 |
Deprotection of benzaldehyde diacetates by ceric ammonium nitrate coated on silica P Cotelle, JP Catteau Tetrahedron letters 33 (27), 3855-3858, 1992 | 70 | 1992 |
Dichlorolissoclimide, a new cytotoxic labdane derivative from Lissoclinum voeltzkowiMichaelson (Urochordata) C Malochet-Grivois, P Cotelle, JF Biard, JP Hénichart, C Debitus, ... Tetrahedron letters 32 (46), 6701-6702, 1991 | 66 | 1991 |
Spectroscopic studies of diketoacids− metal interactions. A probing tool for the pharmacophoric intermetallic distance in the HIV-1 integrase active site C Maurin, F Bailly, E Buisine, H Vezin, G Mbemba, JF Mouscadet, ... Journal of medicinal chemistry 47 (22), 5583-5586, 2004 | 61 | 2004 |
Inhibition of hepatitis B virus replication by N-hydroxyisoquinolinediones and related polyoxygenated heterocycles TC Edwards, E Lomonosova, JA Patel, Q Li, JA Villa, AK Gupta, ... Antiviral research 143, 205-217, 2017 | 59 | 2017 |