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Cited by
Year
Methods and protocols of modern solid phase peptide synthesis
M Amblard, JA Fehrentz, J Martinez, G Subra
Molecular biotechnology 33, 239-254, 2006
7442006
An efficient synthesis of optically active α-(t-butoxycarbonylamino)-aldehydes from α-amino acids
JA Fehrentz, B Castro
Synthesis 1983 (08), 676-678, 1983
3611983
Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons
M Schaeffer, F Langlet, C Lafont, F Molino, DJ Hodson, T Roux, ...
Proceedings of the National Academy of Sciences 110 (4), 1512-1517, 2013
3022013
Synthesis of 3, 4, 5-Trisubstituted-1, 2, 4-triazoles
A Moulin, M Bibian, AL Blayo, S El Habnouni, J Martinez, JA Fehrentz
Chemical reviews 110 (4), 1809-1827, 2010
2022010
High constitutive activity is an intrinsic feature of ghrelin receptor protein
M Damian, J Marie, JP Leyris, JA Fehrentz, P Verdie, J Martinez, ...
Journal of biological chemistry 287 (6), 3630-3641, 2012
1642012
Palatability can drive feeding independent of AgRP neurons
RGP Denis, A Joly-Amado, E Webber, F Langlet, M Schaeffer, SL Padilla, ...
Cell metabolism 22 (4), 646-657, 2015
1502015
Toward potent ghrelin receptor ligands based on trisubstituted 1, 2, 4-triazole structure. 2. Synthesis and pharmacological in vitro and in vivo evaluations
A Moulin, L Demange, G Bergé, D Gagne, J Ryan, D Mousseaux, A Heitz, ...
Journal of medicinal chemistry 50 (23), 5790-5806, 2007
1452007
Solid phase synthesis of chiral 3-substituted quinazoline-2, 4-diones
L Gouilleux, JA Fehrentz, F Winternitz, J Martinez
Tetrahedron letters 37 (39), 7031-7034, 1996
1271996
Ligands and signaling proteins govern the conformational landscape explored by a G protein-coupled receptor
S Mary, M Damian, M Louet, N Floquet, JA Fehrentz, J Marie, J Martinez, ...
Proceedings of the National Academy of Sciences 109 (21), 8304-8309, 2012
1182012
Synthesis and pharmacological in vitro and in vivo evaluations of novel triazole derivatives as ligands of the ghrelin receptor. 1
L Demange, D Boeglin, A Moulin, D Mousseaux, J Ryan, G Bergé, ...
Journal of medicinal chemistry 50 (8), 1939-1957, 2007
1182007
N-terminal liver-expressed antimicrobial peptide 2 (LEAP2) region exhibits inverse agonist activity toward the ghrelin receptor
C M’Kadmi, A Cabral, F Barrile, J Giribaldi, S Cantel, M Damian, S Mary, ...
Journal of Medicinal Chemistry 62 (2), 965-973, 2018
1162018
Improved solid phase synthesis of C-terminal peptide aldehydes
JA Fehrentz, M Paris, A Heitz, J Velek, CF Liu, F Winternitz, J Martinez
Tetrahedron letters 36 (43), 7871-7874, 1995
1121995
Detergent-free isolation of functional G protein-coupled receptors into nanometric lipid particles
C Logez, M Damian, C Legros, C Dupré, M Guéry, S Mary, R Wagner, ...
Biochemistry 55 (1), 38-48, 2016
1092016
New active series of growth hormone secretagogues
V Guerlavais, D Boeglin, D Mousseaux, C Oiry, A Heitz, R Deghenghi, ...
Journal of medicinal chemistry 46 (7), 1191-1203, 2003
962003
Agonism, antagonism, and inverse agonism bias at the ghrelin receptor signaling
C M'Kadmi, JP Leyris, L Onfroy, C Galés, A Saulière, D Gagne, M Damian, ...
Journal of Biological Chemistry 290 (45), 27021-27039, 2015
922015
Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a
JP Leyris, T Roux, E Trinquet, P Verdié, JA Fehrentz, N Oueslati, ...
Analytical biochemistry 408 (2), 253-262, 2011
912011
Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor: Gq complex
M Damian, S Mary, M Maingot, C M'Kadmi, D Gagne, JP Leyris, ...
Proceedings of the National Academy of Sciences 112 (5), 1601-1606, 2015
892015
Ghrelin stimulation of growth hormone-releasing hormone neurons is direct in the arcuate nucleus
G Osterstock, P Escobar, V Mitutsova, LA Gouty-Colomer, P Fontanaud, ...
PLoS One 5 (2), e9159, 2010
892010
Regulation of ERK1/2 activity by ghrelin‐activated growth hormone secretagogue receptor 1A involves a PLC/PKCɛ pathway
D Mousseaux, L Le Gallic, J Ryan, C Oiry, D Gagne, JA Fehrentz, ...
British journal of pharmacology 148 (3), 350-365, 2006
892006
Solution and solid-supported synthesis of 3, 4, 5-trisubstituted 1, 2, 4-triazole-based peptidomimetics
D Boeglin, S Cantel, A Heitz, J Martinez, JA Fehrentz
Organic letters 5 (23), 4465-4468, 2003
862003
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