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Mostafa M. Elbadawi
Mostafa M. Elbadawi
Assistant Professor, Pharmaceutical Chemistry, Kafrelsheikh University
Verified email at pharm.kfs.edu.eg - Homepage
Title
Cited by
Cited by
Year
Discovery of 4-alkoxy-2-aryl-6, 7-dimethoxyquinolines as a new class of topoisomerase I inhibitors endowed with potent in vitro anticancer activity
MM Elbadawi, WM Eldehna, W Wang, KK Agama, Y Pommier, M Abe
European journal of medicinal chemistry 215, 113261, 2021
292021
Design and synthesis of benzothiazole-based SLC-0111 analogues as new inhibitors for the cancer-associated carbonic anhydrase isoforms IX and XII
T Al-Warhi, MM Elbadawi, A Bonardi, A Nocentini, AA Al-Karmalawy, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 2635-2643, 2022
252022
Identification of N-phenyl-2-(phenylsulfonyl) acetamides/propanamides as new SLC-0111 analogues: synthesis and evaluation of the carbonic anhydrase inhibitory activities
MM Elbadawi, WM Eldehna, A Nocentini, MF Abo-Ashour, EB Elkaeed, ...
European Journal of Medicinal Chemistry 218, 113360, 2021
252021
Discovery of 2, 4-thiazolidinedione-tethered coumarins as novel selective inhibitors for carbonic anhydrase IX and XII isoforms
WM Eldehna, MS Taghour, T Al-Warhi, A Nocentini, MM Elbadawi, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 531-541, 2022
172022
2-Arylquinolines as novel anticancer agents with dual EGFR/FAK kinase inhibitory activity: synthesis, biological evaluation, and molecular modelling insights
MM Elbadawi, WM Eldehna, AA Abd El-Hafeez, WR Somaa, A Albohy, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 355-378, 2022
162022
Development of 4-((3-oxo-3-phenylpropyl) amino) benzenesulfonamide derivatives utilizing tail/dual-tail approaches as novel carbonic anhydrase inhibitors
MM Elbadawi, WM Eldehna, A Nocentini, WR Somaa, ST Al-Rashood, ...
European Journal of Medicinal Chemistry 238, 114412, 2022
162022
Design, synthesis and biological evaluation of novel thiohydantoin derivatives as antiproliferative agents: A combined experimental and theoretical assessments
MM Elbadawi, AI Khodair, MK Awad, SE Kassab, MT Elsaady, ...
Journal of Molecular Structure 1249, 131574, 2022
162022
Design, synthesis, molecular docking and cytotoxicity evaluation of some novel 5-arylidene-3-(substituted phenyl)-2-(p-tolylamino)-4-imidazolones
AI Khodair, MM Elbadawi, MT Elsaady, KRA Abdellatif
Journal of Applied Pharmaceutical Science 7 (9), 058-068, 2017
162017
Design, synthesis and cytotoxicity evaluation of new 3, 5-disubstituted-2-thioxoimidazolidinones
KRA Abdellatif, MM Elbadawi, MT Elsaady, AA Abd El-Hafeez, T Fujimura, ...
Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2018
152018
Discovery of indolinone-bearing benzenesulfonamides as new dual carbonic anhydrase and VEGFR-2 inhibitors possessing anticancer and pro-apoptotic properties
S Saied, M Shaldam, MM Elbadawi, S Giovannuzzi, A Nocentini, ...
European Journal of Medicinal Chemistry 259, 115707, 2023
82023
Design and synthesis of 6-arylpyridine-tethered sulfonamides as novel selective inhibitors of carbonic anhydrase IX with promising antitumor features toward the human …
WM Eldehna, EE Mohammed, GH Al-Ansary, E Berrino, MM Elbadawi, ...
European Journal of Medicinal Chemistry 258, 115538, 2023
72023
1, 5-diaryl-1, 2, 4-triazole ureas as new SLC-0111 analogues endowed with dual carbonic anhydrase and VEGFR-2 inhibitory activities
AE Elsawi, MM Elbadawi, A Nocentini, H Almahli, S Giovannuzzi, ...
Journal of Medicinal Chemistry 66 (15), 10558-10578, 2023
62023
Development of new thiazolidine-2, 4-dione hybrids as aldose reductase inhibitors endowed with antihyperglycaemic activity: design, synthesis, biological investigations, and in …
A Hamdi, M Yaseen, WA Ewes, MA Bhat, NI Ziedan, HW El-Shafey, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2231170, 2023
32023
Design, synthesis and biological evaluation of novel quinoline based small molecules as anticancer agents targeting topoisomerase Ⅰ
MMM Elbadawi
広島大学, 2021
2021
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Articles 1–14