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Alessio Nocentini
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Benzothiazole derivatives as anticancer agents
A Irfan, F Batool, SA Zahra Naqvi, A Islam, SM Osman, A Nocentini, ...
Journal of enzyme inhibition and medicinal chemistry 35 (1), 265-279, 2020
1972020
Carbonic anhydrase inhibitors as antitumor/antimetastatic agents: a patent review (2008–2018)
A Nocentini, CT Supuran
Expert Opinion on Therapeutic Patents 28 (10), 729-740, 2018
1922018
Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery
A Nocentini, CT Supuran
Expert Opinion on Drug Discovery 14 (11), 1175-1197, 2019
1402019
Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment
A Angeli, F Carta, A Nocentini, JY Winum, R Zalubovskis, A Akdemir, ...
Metabolites 10 (10), 412, 2020
1282020
Novel 4/3-((4-oxo-5-(2-oxoindolin-3-ylidene) thiazolidin-2-ylidene) amino) benzenesulfonamides: Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and …
WM Eldehna, MF Abo-Ashour, A Nocentini, P Gratteri, IH Eissa, M Fares, ...
European journal of medicinal chemistry 139, 250-262, 2017
1272017
Benzoxaborole compounds for therapeutic uses: a patent review (2010-2018)
A Nocentini, CT Supuran, JY Winum
Expert opinion on therapeutic patents 28 (6), 493-504, 2018
1102018
Benzenesulfonamides incorporating flexible triazole moieties are highly effective carbonic anhydrase inhibitors: synthesis and kinetic, crystallographic, computational, and …
A Nocentini, M Ferraroni, F Carta, M Ceruso, P Gratteri, C Lanzi, E Masini, ...
Journal of Medicinal Chemistry 59 (23), 10692-10704, 2016
1002016
Bacterial ι-carbonic anhydrase: a new active class of carbonic anhydrase identified in the genome of the Gram-negative bacterium Burkholderia territorii
S Del Prete, A Nocentini, CT Supuran, C Capasso
Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 1060-1068, 2020
932020
Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII
A Nocentini, F Carta, M Ceruso, G Bartolucci, CT Supuran
Bioorganic & Medicinal Chemistry 23 (21), 6955-6966, 2015
902015
Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase
A Nocentini, A Angeli, F Carta, JY Winum, R Zalubovskis, S Carradori, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 36 (1), 561-580, 2021
892021
Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC …
WM Eldehna, MF Abo-Ashour, A Nocentini, RS El-Haggar, S Bua, ...
European journal of medicinal chemistry 162, 147-160, 2019
892019
Sulfonamide inhibitors of human carbonic anhydrases designed through a three-tails approach: improving ligand/isoform matching and selectivity of action
A Bonardi, A Nocentini, S Bua, J Combs, C Lomelino, J Andring, ...
Journal of medicinal chemistry 63 (13), 7422-7444, 2020
862020
An overview on the recently discovered iota-carbonic anhydrases
A Nocentini, CT Supuran, C Capasso
Journal of Enzyme Inhibition and Medicinal Chemistry 36 (1), 1988-1995, 2021
822021
Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms
A Nocentini, A Bonardi, P Gratteri, B Cerra, A Gioiello, CT Supuran
Journal of Enzyme Inhibition and Medicinal Chemistry 33 (1), 1453-1459, 2018
812018
Continued exploration of 1, 2, 4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX …
M Krasavin, A Shetnev, T Sharonova, S Baykov, S Kalinin, A Nocentini, ...
European Journal of Medicinal Chemistry 164, 92-105, 2019
802019
3-Hydrazinoisatin-based benzenesulfonamides as novel carbonic anhydrase inhibitors endowed with anticancer activity: Synthesis, in vitro biological evaluation and in silico …
MF Abo-Ashour, WM Eldehna, A Nocentini, A Bonardi, S Bua, HS Ibrahim, ...
European Journal of Medicinal Chemistry 184, 111768, 2019
742019
A new kid on the block? Carbonic anhydrases as possible new targets in Alzheimer’s disease
G Provensi, F Carta, A Nocentini, CT Supuran, F Casamenti, MB Passani, ...
International journal of molecular sciences 20 (19), 4724, 2019
722019
Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer
WM Eldehna, A Nocentini, ST Al-Rashood, GS Hassan, HM Alkahtani, ...
Bioorganic Chemistry 81, 425-432, 2018
702018
Selenols: A new class of carbonic anhydrase inhibitors
A Angeli, D Tanini, A Nocentini, A Capperucci, M Ferraroni, P Gratteri, ...
Chemical communications 55 (5), 648-651, 2019
682019
Deciphering the mechanism of human carbonic anhydrases inhibition with sulfocoumarins: computational and experimental studies
A Nocentini, F Carta, M Tanc, S Selleri, CT Supuran, C Bazzicalupi, ...
Chemistry–A European Journal 24 (31), 7840-7844, 2018
672018
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