Ghada S. Hassan
Ghada S. Hassan
Professor of Medicinal Chemistry
Verified email at mans.edu.eg - Homepage
TitleCited byYear
Substituted thiazoles V. Synthesis and antitumor activity of novel thiazolo [2, 3-b] quinazoline and pyrido [4, 3-d] thiazolo [3, 2-a] pyrimidine analogues
FAM Al-Omary, GS Hassan, SM El-Messery, HI El-Subbagh
European journal of medicinal chemistry 47, 65-72, 2012
832012
Substituted thiazoles VII. Synthesis and antitumor activity of certain 2-(substituted amino)-4-phenyl-1, 3-thiazole analogs
GS Hassan, SM El-Messery, FAM Al-Omary, HI El-Subbagh
Bioorganic & medicinal chemistry letters 22 (20), 6318-6323, 2012
562012
Synthesis and biological evaluation of some polymethoxylated fused pyridine ring systems as antitumor agents
SAF Rostom, GS Hassan, HI El‐Subbagh
Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2009
552009
Substituted thiazoles VI. Synthesis and antitumor activity of new 2-acetamido-and 2 or 3-propanamido-thiazole analogs
SM El-Messery, GS Hassan, FAM Al-Omary, HI El-Subbagh
European journal of medicinal chemistry 54, 615-625, 2012
542012
Nonclassical antifolates, Part 4. 5-(2-Aminothiazol-4-yl)-4-phenyl-4H-1,2,4-triazole-3-thiols as a new class of DHFR inhibitors: Synthesis, biological evaluation and molecular …
HIES Ghada S. Hassan, Shahenda M. El-Messery, Fatmah A
European Journal of Medicinal Chemistry, 2013
402013
Nonclassical antifolates, part 3: synthesis, biological evaluation and molecular modeling study of some new 2-heteroarylthio-quinazolin-4-ones
FAM Al-Omary, GS Hassan, SM El-Messery, MN Nagi, ESE Habib, ...
European journal of medicinal chemistry 63, 33-45, 2013
382013
Nonclassical antifolates, part 5. Benzodiazepine analogs as a new class of DHFR inhibitors: Synthesis, antitumor testing and molecular modeling study
HI El-Subbagh, GS Hassan, SM El-Messery, ST Al-Rashood, ...
European journal of medicinal chemistry 74, 234-245, 2014
312014
Novel 4(3H)-quinazolinone analogs: synthesis and anticonvulsant
AS El-Azab, SG Abdel-Hamide, MM Sayed-Ahmed, GS Hassan, ...
Medicinal Chemistry Research 22 (6), 2815-2827, 2013
312013
Synthesis and anticonvulsant activity of some new thiazolo [3, 2-a][1, 3] diazepine, benzo [d] thiazolo [5, 2-a][12, 6] diazepine and benzo [d] oxazolo [5, 2-a][12, 6 …
HI El-Subbagh, GS Hassan, AS El-Azab, AM Alaa, AA Kadi, AM Al-Obaid, ...
European journal of medicinal chemistry 46 (11), 5567-5572, 2011
242011
Synthesis, biological evaluation and molecular modeling study of 2-(1, 3, 4-thiadiazolyl-thio and 4-methyl-thiazolyl-thio)-quinazolin-4-ones as a new class of DHFR inhibitors
ST Al-Rashood, GS Hassan, SM El-Messery, MN Nagi, ESE Habib, ...
Bioorganic & medicinal chemistry letters 24 (18), 4557-4567, 2014
202014
Synthesis, antimicrobial and antiviral testing of some new 1-adamantyl analogues
AEMB Ghada S. Hassan, Ali A. El-Emam, Laila M. Gad
Saudi Pharmaceutical Journal 18, 123-128, 2010
182010
Synthesis, biological evaluation and molecular modeling study of new (1, 2, 4-triazole or 1, 3, 4-thiadiazole)-methylthio-derivatives of quinazolin-4 (3H)-one as DHFR inhibitors
YI El-Gazzar, HH Georgey, SM El-Messery, HA Ewida, GS Hassan, ...
Bioorganic chemistry 72, 282-292, 2017
142017
Menadione
GS Hassan
Profiles of Drug Substances, Excipients, and Related Methodology 38, 227-313, 2013
142013
Synthesis and anticancer activity of new thiazolo [3, 2-a] pyrimidines: DNA binding and molecular modeling study
GS Hassan, SM El-Messery, A Abbas
Bioorganic chemistry 74, 41-52, 2017
132017
Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer
WM Eldehna, A Nocentini, ST Al-Rashood, GS Hassan, HM Alkahtani, ...
Bioorganic chemistry 81, 425-432, 2018
122018
Synthesis and antitumor activity of certain new thiazolo[2,3-b]quinazoline and thiazolo[3,2-a]pyrimidine analogs
GS Hassan
Medicinal Chemistry Research, 2013
112013
New ultra-short acting hypnotic: Synthesis, biological evaluation, and metabolic profile of ethyl 8-oxo-5, 6, 7, 8-tetrahydro-thiazolo [3, 2-a][1, 3] diazepin-3-carboxylate …
HI El-Subbagh, HA El-Kashef, AA Kadi, AM Alaa, GS Hassan, J Tettey, ...
Bioorganic & medicinal chemistry letters 18 (1), 72-77, 2008
112008
Synthesis, Ultra‐Short Acting Hypnotic Activity, and Metabolic Profile of Ethyl 8‐Oxo‐5,6,7,8‐tetrahydro‐thiazolo[3,2‐a] [1,3]diazepin‐3‐carboxylate (HIE‐124)
AA Kadi, HA El‐Kashef, AAM Abdel‐Aziz, GS Hassan, J Tettey, MH Grant, ...
Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2008
102008
Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC …
WM Eldehna, MF Abo-Ashour, A Nocentini, RS El-Haggar, S Bua, ...
European journal of medicinal chemistry 162, 147-160, 2019
92019
SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX
WM Eldehna, MF Abo-Ashour, E Berrino, D Vullo, HA Ghabbour, ...
Bioorganic chemistry 83, 549-558, 2019
82019
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